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Machine translation
1. (WO1997019911) AMINO ACID DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS AND PROCESSES FOR PREPARING THEM
Latest bibliographic data on file with the International Bureau   

Pub. No.:    WO/1997/019911    International Application No.:    PCT/EP1996/005222
Publication Date: 05.06.1997 International Filing Date: 26.11.1996
Chapter 2 Demand Filed:    16.04.1997    
IPC:
A61K 38/00 (2006.01), C07C 257/18 (2006.01), C07C 275/24 (2006.01), C07C 275/56 (2006.01), C07C 279/14 (2006.01), C07C 279/24 (2006.01), C07C 279/36 (2006.01), C07C 307/06 (2006.01), C07C 311/35 (2006.01), C07D 209/08 (2006.01), C07D 209/18 (2006.01), C07D 209/24 (2006.01), C07D 209/42 (2006.01), C07D 209/44 (2006.01), C07D 223/20 (2006.01), C07D 233/26 (2006.01), C07D 233/36 (2006.01), C07D 233/72 (2006.01), C07D 233/88 (2006.01), C07D 235/06 (2006.01), C07D 235/08 (2006.01), C07D 239/46 (2006.01), C07D 249/14 (2006.01), C07D 271/06 (2006.01), C07D 307/85 (2006.01), C07K 5/078 (2006.01)
Applicants: DR. KARL THOMAE GMBH [DE/DE]; Patentstelle, Birkendorfer Strasse 65, D-88397 Biberach (DE) (For All Designated States Except US).
ENGEL, Wolfhard [DE/DE]; (DE) (For US Only).
EBERLEIN, Wolfgang [DE/DE]; (DE) (For US Only).
RUDOLF, Klaus [DE/DE]; (DE) (For US Only).
DOODS, Henri [NL/DE]; (DE) (For US Only).
WIELAND, Heike-Andrea [DE/DE]; (DE) (For US Only).
WILLIM, Klaus-Dieter [DE/DE]; (DE) (For US Only).
ENTZEROTH, Michael [DE/DE]; (DE) (For US Only).
WIENEN, Wolfgang [DE/DE]; (DE) (For US Only)
Inventors: ENGEL, Wolfhard; (DE).
EBERLEIN, Wolfgang; (DE).
RUDOLF, Klaus; (DE).
DOODS, Henri; (DE).
WIELAND, Heike-Andrea; (DE).
WILLIM, Klaus-Dieter; (DE).
ENTZEROTH, Michael; (DE).
WIENEN, Wolfgang; (DE)
Priority Data:
195 44 687.9 30.11.1995 DE
Title (EN) AMINO ACID DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS AND PROCESSES FOR PREPARING THEM
(FR) DERIVES D'ACIDES AMINES, COMPOSITIONS PHARMACEUTIQUES CONTENANT CES COMPOSES ET PROCEDES DE PREPARATION DE CEUX-CI
Abstract: front page image
(EN)The invention relates to new amino acid derivatives of general formula (I), wherein B, T, Z, Y, V and n are defined as in claim 1, the tautomers, diastereomers and enantiomers thereof, the mixtures thereof and the salts thereof, particularly their physiologically acceptable salts with inorganic or organic acids or bases which have valuable pharmacological properties, particularly selective NPY-antagonist properties, pharmaceutical compositions containing these compounds, the use thereof and processes for preparing them.
(FR)L'invention concerne des nouveaux dérivés d'acides aminés de la formule générale (I), dans laquelle B, T, Z, Y, V et n sont tels que définis dans la revendication 1. L'invention concerne également des tautomères, diastéréomères et énantiomères de ces dérivés et leurs mélanges, ainsi que des sels de ces dérivés, notamment des sels d'addition d'acides ou de bases inorganiques ou organiques, acceptables sur le plan physiologique. Ces dérivés possèdent des propriétés pharmacologiques précieuses, notamment des propriétés antagonistes du neuropeptide Y. On décrit encore des compositions pharmaceutiques contenant ces composés ainsi que l'utilisation et des procédés de préparation de celles-ci.
Designated States: CA, JP, MX, US.
European Patent Office (AT, BE, CH, DE, DK, ES, FI, FR, GB, GR, IE, IT, LU, MC, NL, PT, SE).
Publication Language: English (EN)
Filing Language: English (EN)