Some content of this application is unavailable at the moment.
If this situation persists, please contact us atFeedback&Contact
1. (WO1997015571) METHOD FOR TREATING CANCER USING TAXOID ONIUM SALT PRODRUGS
Latest bibliographic data on file with the International Bureau

Pub. No.: WO/1997/015571 International Application No.: PCT/US1995/013902
Publication Date: 01.05.1997 International Filing Date: 27.10.1995
Chapter 2 Demand Filed: 22.05.1997
IPC:
A61K 31/337 (2006.01) ,A61K 31/381 (2006.01) ,A61K 31/4427 (2006.01) ,C07D 405/12 (2006.01)
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
K
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31
Medicinal preparations containing organic active ingredients
33
Heterocyclic compounds
335
having oxygen as the only ring hetero atom, e.g. fungichromin
337
having four-membered rings, e.g. taxol
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
K
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31
Medicinal preparations containing organic active ingredients
33
Heterocyclic compounds
38
having sulfur as a ring hetero atom
381
having five-membered rings
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
K
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31
Medicinal preparations containing organic active ingredients
33
Heterocyclic compounds
395
having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins
435
having six-membered rings with one nitrogen as the only ring hetero atom
44
Non-condensed pyridines; Hydrogenated derivatives thereof
4427
containing further heterocyclic ring systems
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
D
HETEROCYCLIC COMPOUNDS
405
Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
02
containing two hetero rings
12
linked by a chain containing hetero atoms as chain links
Applicants:
THE SCRIPPS RESEARCH INSTITUTE [US/US]; 10550 North Torrey Pines Road La Jolla, CA 92037, US (AllExceptUS)
WRASIDLO, Wolfgang [DE/DE]; DE (UsOnly)
Inventors:
WRASIDLO, Wolfgang; DE
Agent:
LEWIS, Donald, G. ; The Scripps Research Institute 10550 North Torrey Pines Road, TPC-8 La Jolla, CA 92037, US
Priority Data:
Title (EN) METHOD FOR TREATING CANCER USING TAXOID ONIUM SALT PRODRUGS
(FR) PROCEDE DE TRAITEMENT DU CANCER AU MOYEN DE PROMEDICAMENTS A BASE DE SELS D'ONIUM TAXOÏDES
Abstract:
(EN) C-2'-methylpyridinium acetates (MPA)-taxol and C-2'-methylpyridinium acetates (MPA)-taxotere are prodrugs having good aqueous solubility, low toxicity and high anti-tumor activity. These prodrugs are administered to patients for treating tumors. Administration may be by injection or infusion.
(FR) Les acétates de C-2'-méthylpyridinium (MPA)-taxotère sont des promédicaments ayant une bonne solubilité aqueuse, une faible toxicité et une haute activité antitumorale. Ces promédicaments sont administrés à des patients afin de traiter des tumeurs. Cette administration peut se faire par injection ou perfusion.
Designated States: AL, AM, AT, AU, BB, BG, BR, BY, CA, CH, CN, CZ, DE, DK, EE, ES, FI, GB, GE, HU, IS, JP, KE, KG, KP, KR, KZ, LK, LR, LS, LT, LU, LV, MD, MG, MK, MN, MW, MX, NO, NZ, PL, PT, RO, RU, SD, SE, SG, SI, SK, TJ, TM, TT, UA, UG, US, UZ, VN
African Regional Intellectual Property Organization (ARIPO) (KE, LS, MW, SD, SZ, UG)
European Patent Office (AT, BE, CH, DE, DK, ES, FR, GB, GR, IE, IT, LU, MC, NL, PT, SE)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, ML, MR, NE, SN, TD, TG)
Publication Language: English (EN)
Filing Language: English (EN)
Also published as:
AU1995040135