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1. WO1996011931 - POLYCYCLIC FUSED RING MODULATORS OF ACETYLCHOLINE RECEPTORS

Publication Number WO/1996/011931
Publication Date 25.04.1996
International Application No. PCT/US1995/012905
International Filing Date 28.09.1995
Chapter 2 Demand Filed 09.05.1996
IPC
C07D 471/04 2006.01
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
471Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/-C07D463/251
02in which the condensed system contains two hetero rings
04Ortho-condensed systems
C07D 491/14 2006.01
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
491Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/-C07D459/290
12in which the condensed system contains three hetero rings
14Ortho-condensed systems
CPC
C07D 471/04
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
471Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
02in which the condensed system contains two hetero rings
04Ortho-condensed systems
C07D 491/14
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
491Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
12in which the condensed system contains three hetero rings
14Ortho-condensed systems
Applicants
  • SIBIA NEUROSCIENCES, INC. [US]/[US] (AllExceptUS)
  • WHITTEN, Jeffrey, P. [GB]/[US] (UsOnly)
  • MCDONALD, Ian, A. [AU]/[US] (UsOnly)
  • VERNIER, Jean-Michel [FR]/[US] (UsOnly)
Inventors
  • WHITTEN, Jeffrey, P.
  • MCDONALD, Ian, A.
  • VERNIER, Jean-Michel
Agents
  • REITER, Stephen, E.
  • FIENER, Josef
Priority Data
08/322,75713.10.1994US
Publication Language English (EN)
Filing Language English (EN)
Designated States
Title
(EN) POLYCYCLIC FUSED RING MODULATORS OF ACETYLCHOLINE RECEPTORS
(FR) MODULATEURS POLYCYCLIQUES A NOYAU FUSIONNE DE RECEPTEURS D'ACETYLCHOLINE
Abstract
(EN)
In accordance with the present invention, there is provided a class of polycyclic fused ring compounds of formula (I) which are modulators of acetylcholine receptors. The compounds of the invention displace acetylcholine receptor ligands from their binding sites. Invention compounds may act as agonists, partial agonists, antagonists or allosteric modulators of acetylcholine receptors.
(FR)
La présente invention se rapporte à une classe de composés polycycliques à noyau fusionné de la formule (I), agissant comme modulateurs des récepteurs d'acétylcholine. Les composés selon la présente invention déplacent les ligands des récepteurs d'acétylcholine de leurs sites de liaison. Ils peuvent agir comme agonistes, agonistes partiels, antagonistes ou modulateurs allostériques des récepteurs d'acétylcholine.
Also published as
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