Processing

Please wait...

Settings

Settings

1. WO1996005200 - TETRAHYDROPYRIDINYLMETHYL DERIVATIVES OF PYRROLO[2,3-b]PYRIDINE

Publication Number WO/1996/005200
Publication Date 22.02.1996
International Application No. PCT/GB1995/001820
International Filing Date 01.08.1995
Chapter 2 Demand Filed 17.01.1996
IPC
C07D 471/04 2006.01
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
471Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/-C07D463/251
02in which the condensed system contains two hetero rings
04Ortho-condensed systems
CPC
C07D 471/04
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
471Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
02in which the condensed system contains two hetero rings
04Ortho-condensed systems
Applicants
  • MERCK SHARP & DOHME LIMITED [GB/GB]; Hertford Road Hoddesdon Hertfordshire EN11 9BU, GB (AllExceptUS)
  • CURTIS, Neil, Roy [GB/GB]; GB (UsOnly)
  • KULAGOWSKI, Janusz, Jozef [GB/GB]; GB (UsOnly)
  • LEESON, Paul, David [GB/US]; GB (UsOnly)
  • RIDGILL, Mark, Peter [GB/GB]; GB (UsOnly)
Inventors
  • CURTIS, Neil, Roy; GB
  • KULAGOWSKI, Janusz, Jozef; GB
  • LEESON, Paul, David; GB
  • RIDGILL, Mark, Peter; GB
Agents
  • THOMPSON, John; Merck & Co., Inc. European Patent Dept. Terlings Park, Eastwick Road Harlow Essex CM20 2QR, GB
Priority Data
9416160.110.08.1994GB
9416161.910.08.1994GB
9505888.923.03.1995GB
Publication Language English (EN)
Filing Language English (EN)
Designated States
Title
(EN) TETRAHYDROPYRIDINYLMETHYL DERIVATIVES OF PYRROLO[2,3-b]PYRIDINE
(FR) DERIVES TETRAHYDROPYRIDINYLMETHYLE DE PYRROLO[2,3-b]PYRIDINE
Abstract
(EN)
A class of pyrrolo[2,3-b]pyridine derivatives of formula (I), wherein Q represents a moiety of formula Qa or Qb, are ligands for dopamine receptor subtypes within the body, in particular the dopamine D4 receptor subtype and are therefore useful in the treatment and/or prevention of disorders of the dopamine system, including schizophrenia.
(FR)
Classe de dérivés de pyrrolo[2,3-b]pyridine, de la formule (I), dans laquelle Q représente une fraction de formule Qa ou Qb. Ces dérivés sont des ligands de sous-types de récepteurs de la dopamine dans le corps, notamment du sous-type de récepteur D4 de la dopamine, et ils sont par conséquent utiles dans le traitement et/ou la prévention de troubles du système dopamine, notamment de la schizophrénie.
Latest bibliographic data on file with the International Bureau