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1. WO1996002509 - QUINOLINE DERIVATIVES AS NK¿3? ANTAGONISTS

Publication Number WO/1996/002509
Publication Date 01.02.1996
International Application No. PCT/EP1995/002638
International Filing Date 06.07.1995
Chapter 2 Demand Filed 20.01.1996
IPC
C07D 215/20 2006.01
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
215Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
02having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
16with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
20Oxygen atoms
C07D 215/52 2006.01
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
215Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
02having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
16with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
48Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
50attached in position 4
52with aryl radicals attached in position 2
C07D 401/12 2006.01
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
401Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
02containing two hetero rings
12linked by a chain containing hetero atoms as chain links
CPC
C07D 215/20
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
215Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
02having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
16with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
20Oxygen atoms
C07D 215/52
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
215Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
02having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
16with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
48Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
50attached in position 4
52with aryl radicals attached in position 2
C07D 401/12
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
401Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
02containing two hetero rings
12linked by a chain containing hetero atoms as chain links
Applicants
  • SMITHKLINE BEECHAM FARMACEUTICI S.P.A. [IT/IT]; Via Zambeletti I-20021 Baranzate, IT (AllExceptUS)
  • FARINA, Carlo [IT/IT]; IT (UsOnly)
  • GIARDINA, Giuseppe, Arnaldo, Maria [IT/IT]; IT (UsOnly)
  • GRUGNI, Mario [IT/IT]; IT (UsOnly)
  • RAVEGLIA, Luca, Francesco [IT/IT]; IT (UsOnly)
Inventors
  • FARINA, Carlo; IT
  • GIARDINA, Giuseppe, Arnaldo, Maria; IT
  • GRUGNI, Mario; IT
  • RAVEGLIA, Luca, Francesco; IT
Agents
  • RUSSELL, Brian, John; SmithKline Beecham Corporate Intellectual Property SB House, Great West Road Brentford Middlesex TW8 9BD, GB
  • GIDDINGS, Peter, John; SmithKline Beecham Corporate Intellectual Property SB House, Great West Road Brentford, Middlesex TW8 9BD, GB
Priority Data
MI94A00146614.07.1994IT
Publication Language English (EN)
Filing Language English (EN)
Designated States
Title
(EN) QUINOLINE DERIVATIVES AS NK3 ANTAGONISTS
(FR) DERIVES DE QUINOLINE UTILISES COMME ANTAGONISTES DE LA NEUROKININE 3 (NK3)
Abstract
(EN)
NK3 receptor antagonists of formula (I) are useful in the treatment of pulmonary and CNS disorders.
(FR)
Des antagonistes du récepteur de NK3 de la formule (I) conviennent au traitement de troubles pulmonaires et du système nerveux central.
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