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Machine translation
1. (WO1994026702) N-ACYL SULFAMIC ACID ESTERS (OR THIOESTERS), N-ACYL SULFONAMIDES, AND N-SULFONYL CARBAMIC ACID ESTERS (OR THIOESTERS) AS HYPERCHOLESTEROLEMIC AGENTS
Latest bibliographic data on file with the International Bureau   

Pub. No.:    WO/1994/026702    International Application No.:    PCT/US1994/005233
Publication Date: 24.11.1994 International Filing Date: 11.05.1994
Chapter 2 Demand Filed:    01.12.1994    
IPC:
A61K 31/18 (2006.01), C07C 307/02 (2006.01), C07C 311/51 (2006.01), C07D 311/84 (2006.01)
Applicants: WARNER-LAMBERT COMPANY [US/US]; 2800 Plymouth Road, Ann Arbor, MI 48105 (US)
Inventors: LEE, Helen, Tsenwhei; (US).
PICARD, Joseph, Armand; (US).
SLISKOVIC, Drago, Robert; (US).
WIERENGA, Wendell; (US)
Agent: ANDERSON, Elizabeth, M.; Warner-Lambert Company, 2800 Plymouth Road, Ann Arbor, MI 48105 (US).
MANSMANN, Ivo; Warner-Lambert Company, Legal Division, Patent Department, Gödecke AG, D-79090 Freiburg (DE)
Priority Data:
08/062,515 14.05.1993 US
08/223,932 13.04.1994 US
Title (EN) N-ACYL SULFAMIC ACID ESTERS (OR THIOESTERS), N-ACYL SULFONAMIDES, AND N-SULFONYL CARBAMIC ACID ESTERS (OR THIOESTERS) AS HYPERCHOLESTEROLEMIC AGENTS
(FR) ESTERS (OU THIOESTERS) D'ACIDE N-ACYL SULFAMIQUE, N-ACYL SULFONAMIDES ET ESTERS (OU THIOESTERS) DE L'ACIDE N-SULFONYL CARBAMIQUE UTILISES COMME AGENTS HYPERCHOLESTEROLEMIQUES
Abstract: front page image
(EN)The present invention is directed to compounds useful for the regulation of cholesterol of formula (I), methods for using them and pharmaceutical compositions thereof. In Formula (I) X and Y are oxgen, sulfur, or (CR'R')¿n? wherein n is 1 to 4; R is hydrogen, alkyl, or benzyl; R¿1? and R¿2? are phenyl, substituted phenyl, naphthyl, substituted naphthyl, an aralkyl group, an alkyl chain, adamantyl, or a cycloalkyl group.
(FR)La présente invention concerne des composés de la formule (I) utiles pour la régulation du cholestérol, ainsi que leurs procédés d'utilisation et des compositions pharmaceutiques les contenant. Dans cette formule, X et Y représentent oxygène, soufre ou (CR'R')¿n?, où n est compris entre 1 et 4, R représente hydrogène, alkyle ou benzyle, R¿1? et R¿2? représentent un groupe phényle, phényle substitué, naphtyle, naphtyle substitué, aralkyle, alkyle, adamantyle ou cycloalkyle.
Designated States: AU, CA, CZ, FI, HU, JP, KR, NO, NZ, RU, SK.
European Patent Office (AT, BE, CH, DE, DK, ES, FR, GB, GR, IE, IT, LU, MC, NL, PT, SE).
Publication Language: English (EN)
Filing Language: English (EN)