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Machine translation
1. (WO1992003441) MACROCYCLIC COMPOUNDS
Latest bibliographic data on file with the International Bureau   

Pub. No.:    WO/1992/003441    International Application No.:    PCT/GB1991/001384
Publication Date: 05.03.1992 International Filing Date: 14.08.1991
Chapter 2 Demand Filed:    14.02.1992    
IPC:
C07D 498/22 (2006.01), C07H 19/01 (2006.01)
Applicants: FISONS PLC [GB/GB]; Fison House, Princes Street, Ipswich, Suffolk IP1 1QH (GB) (For All Designated States Except US).
DONALD, David, Keith [GB/GB]; (GB) (For US Only).
FURBER, Mark [GB/GB]; (GB) (For US Only)
Inventors: DONALD, David, Keith; (GB).
FURBER, Mark; (GB)
Agent: WRIGHT, Robert, Gordon, McRae; Fisons plc, 12 Derby Road, Loughborough, Leicestershire LE11 0BB (GB)
Priority Data:
9018196.7 18.08.1990 GB
9102305.1 02.02.1991 GB
Title (EN) MACROCYCLIC COMPOUNDS
(FR) COMPOSES MACROCYCLIQUES
Abstract: front page image
(EN)Compounds of formula (I) are provided, wherein R?1¿ represents OH or OCH¿3?; R?2¿ represents OH or H; R?3¿ represents methyl, ethyl, propyl or allyl; X represents O, (H,OH) or (H,H); m represents 0 or 1; n represents 1 or 2; and pharmaceutically acceptable derivatives thereof; provided that when n is 1, then R?3¿ is allyl or propyl. The compounds are indicated $i(inter alia) as immunosuppressive agents.
(FR)On décrit des composés macrocycliques de la formule (I) où R?1¿ rreprésente OH ou OCH¿3?, R?2¿ représente OH ou H; R?3¿ représente méthyle, éthyle, propyle ou allyle, X représente O, (H,OH) ou (H,H); m vaut 0 ou 1; n vaut 1 ou 2; et des dérivés pharmaceutiquement acceptables de ces éléments; à condition que, lorsque n vaut 1, R?3¿ représente alors allyle ou propyle. Les composés peuvent être utilisés, entre autres, comme agents immunosuppresseurs.
Designated States: AU, BB, BG, BR, CA, CS, FI, HU, JP, KP, KR, LK, MC, MG, MW, NO, PL, RO, SD, SU, US.
European Patent Office (AT, BE, CH, DE, DK, ES, FR, GB, GR, IT, LU, NL, SE).
Publication Language: English (EN)
Filing Language: English (EN)