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1. (WO1985004554) AMIDINE BENZODIAZEPINES, METHODS FOR THEIR USE AND INTERMEDIATES
Latest bibliographic data on file with the International Bureau

Pub. No.: WO/1985/004554 International Application No.: PCT/US1985/000632
Publication Date: 24.10.1985 International Filing Date: 11.04.1985
IPC:
C07D 487/04 (2006.01)
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
D
HETEROCYCLIC COMPOUNDS
487
Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/-C07D477/183
02
in which the condensed system contains two hetero rings
04
Ortho-condensed systems
Applicants:
McNEILAB, INC. [US/US]; Spring House, PA 19477, US
Inventors:
HO, Chih, Yung; US
Agent:
LAMBERT, Benjamin, F.; Johnson & Johnson One Johnson & Johnson Plaza New Brunswick, NJ 08933-7003, US
Priority Data:
599,09511.04.1984US
721,72310.04.1985US
Title (EN) AMIDINE BENZODIAZEPINES, METHODS FOR THEIR USE AND INTERMEDIATES
(FR) BENZODIAZEPINES D'AMIDINE, LEURS PROCEDES D'UTILISATION ET LEURS INTERMEDIAIRES
Abstract:
(EN) Fused tetracyclic benzodiazepines of formula (I), where R1 is an acyclic amine or cyclic amine such as 1-piperidine, 4-morpholine or 1-piperazine and R2 is H or a substituent as defined herein are useful as antiallergins. Also, methods for their synthesis, intermediate used in such synthesis, methods for use as medicaments and pharmaceutical compositions.
(FR) Benzodiazépines tétracycliques fusionnées de formule (I), où R1 est une amine acyclique ou une amine cyclique telle que la 1-pipéridine, la 4-morpholine ou la 1-pipérazine et R2 est H ou un substituant défini. Ces composés sont utiles comme antiallergiques. Sont également décrits des procédés en permettant la synthèse, des intermédiaires utilisés dans cette synthèse, ainsi que des procédés d'utilisation de ces composés dans des médicaments et des compositions pharmaceutiques.
Designated States: AU, DK, JP, KR
European Patent Office (AT, BE, CH, DE, FR, GB, IT, LU, NL, SE)
Publication Language: English (EN)
Filing Language: English (EN)
Also published as:
EP0179128AU1985042333