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Machine translation
1. (WO1982004050) HETEROCYCLIC ALKYLENE TRIAZINONES
Latest bibliographic data on file with the International Bureau   

Pub. No.:    WO/1982/004050    International Application No.:    PCT/US1982/000632
Publication Date: 25.11.1982 International Filing Date: 12.05.1982
IPC:
C07D 251/16 (2006.01), C07D 401/06 (2006.01), C07D 403/06 (2006.01), C07D 405/06 (2006.01), C07D 409/06 (2006.01), C07D 413/06 (2006.01), C07D 417/06 (2006.01), C07D 521/00 (2006.01)
Applicants: RORER INTERNATIONAL (OVERSEAS) INC. [US/US]; 100 West Tenth Street, Wilmington, DE 19899 (US)
Inventors: DOUGLAS, George, Henry; (US).
STUDT, William, Lyon; (US).
WON, Chong, Min; (US).
DODSON, Stuart, Alan; (US).
ZALIPSKY, Jerome, Jaroslaw; (US)
Agent: BARRON, Alexis; Synnestvedt & Lechner, 3131 PSFS Building, 12 South 12th Street, Philadelphia, PA 19107 @ (US)
Priority Data:
262,809 12.05.1981 US
Title (EN) HETEROCYCLIC ALKYLENE TRIAZINONES
(FR) TRIAZINONES D'ALKYLENE HETEROCYCLIQUES
Abstract: front page image
(EN)Heterocyclic alkyl s-triazine compounds are prepared from the corresponding amidinourea and amidinothiourea compounds by reacting with an activated form of an acid amide to give respectively substituted s-triazinones and thiones of the formula (FORMULA) which have pharmacological properties that render them suitable for use for a variety of medicinal purposes, including use as antidiarrheal agents, and which are also useful derivatives in analyzing for the corresponding amidinourea or amidinothiourea precursors.
(FR)Des composes s-triazine d'alkyle heterocycliques sont prepares a partir des composes correspondant d'amidinouree et d'amidinothiouree par reaction avec une forme activee d'une amide acide pour donner respectivement des s-triazinones et thiones substitues de formule (FORMULE) ayant des proprietes pharmacologiques qui les rendent appropries a diverses fins medicinales, y compris leur utilisation comme agents anti-diarrheiques, et sont egalement des derives utiles a l'analyse pour la detection des precurseurs d'amidinouree ou d'amidinothiouree correspondants.
Designated States: AU, JP.
European Patent Office (AT, BE, CH, DE, FR, GB, LU, NL, SE).
Publication Language: English (EN)
Filing Language: English (EN)