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Machine translation
1. (WO1980000152) 3-AMINOPROPOXY-ARYL DERIVATES,PREPARATION AND USE THEREOF
Latest bibliographic data on file with the International Bureau   

Pub. No.:    WO/1980/000152    International Application No.:    PCT/CH1979/000091
Publication Date: 07.02.1980 International Filing Date: 20.06.1979
IPC:
B65B 13/26 (2006.01), C07D 209/08 (2006.01), C07D 209/42 (2006.01)
Applicants:
Inventors:
Priority Data:
7235/78 03.07.1978 CH
Title (EN) 3-AMINOPROPOXY-ARYL DERIVATES,PREPARATION AND USE THEREOF
(FR) DERIVES D"UN 3-AMINOPROPOXY-ARYLE, LEUR PREPARATION ET UTILISATION
Abstract: front page image
(EN)New compounds having the following formula I, (FORMULA) wherein R1 is hydrogen or methyl R3 is hydrogen, methyl, hydroxymethyl, carboxyl, alcoxycarbonyl having 2 to 5 carbon atoms, carbamoyl or cyano and R2 is one of the groups a) to i); these groups are: (FORMULA) and may be used as medicines. These compounds have antiarrhytmic (Alpha)-adrenergic blocking and antihypertension properties; and in case of compounds carrying in position 2 of the indole cycle a cyano or carbamoyl group, (Beta)-adrenergic blocking properties. These compounds are obtained by amination.
(FR)Les nouveaux composes de formule I, (FORMULE) dans laquelle R1, signifie hydrogene ou methyle, R3, signifie hydrogene methyle hydroxymethyle, carboxyle, alcoxycarbonyle avec au total 2 a 5 atomes de carbone, carbamoyle ou cyano et R2 signifie un des groupes a) a i); ces groupes a) a i) signifiant: (FORMULE) peuvent etre utilises comme remede. Ils presentent des proprietes antiarrhytmiques, (Alpha)-adrenergiques bloquantes et antihypertensives; et dans le cas de composes portant en position 2 du cycle indolique un groupement cyano ou carbamoyle, egalement des proprietes (Beta)-adrenergiques bloquantes. L"on obtient ces composes par amination.
Designated States:
Publication Language: German (DE)
Filing Language: German (DE)