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1. TH125651 - SULFAMOYL- PHENYL-UREIDO BENZAMIDINE-DERIVATIVES AS ANTIMALARIAL AGENTS

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Office Thailand
Application Number 1101001339
Application Date 29.01.2010
Publication Number 125651
Publication Date 25.07.2013
Publication Kind A
IPC
C07D 207/09
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
207Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
02with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
04having no double bonds between ring members or between ring members and non-ring members
08with hydrocarbon radicals, substituted by hetero atoms, attached to ring carbon atoms
09Radicals substituted by nitrogen atoms not forming part of a nitro radical
C07D 207/14
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
207Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
02with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
04having no double bonds between ring members or between ring members and non-ring members
10with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
14Nitrogen atoms not forming part of a nitro radical
C07D 209/44
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
209Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
02condensed with one carbocyclic ring
44Iso-indoles; Hydrogenated iso-indoles
C07D 211/22
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
211Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
04with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
06having no double bonds between ring members or between ring members and non-ring members
08with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
18with substituted hydrocarbon radicals attached to ring carbon atoms
20with hydrocarbon radicals, substituted by singly bound oxygen or sulfur atoms
22by oxygen atoms
Applicants 4เอสซี เอจี
Inventors เพกอราโร สเตฟาโน
Agents นายจักรพรรดิ์ มงคลสิทธิ์, นางสาวปรับโยชน์ ศรีกิจจาภรณ์, นายรุทร นพคุณ
Priority Data PCT/EP2010/000546 29.01.2010 -
61/148,617 30.01.2009 US
Title
(EN) SULFAMOYL- PHENYL-UREIDO BENZAMIDINE-DERIVATIVES AS ANTIMALARIAL AGENTS
(TH) อนุพันธ์ซัลฟาโมอิล-เฟนิล-ยูรีอิโด เบนซามีดิน เป็นสารต้านโรคมาลาเรีย
Abstract
(EN)
The present invention relates to novel sulfamoyl-phenyl-ureido compounds having the formula (I) or a physiologically acceptable salt or derivative thereof which are suitable for the therapy of infections caused by protozoa and in particular uncomplicated or severe malaria caused by plasmodia.

(TH)
การประดิษฐ์นี้ เกี่ยวกับ สารประกอบซัลฟา โมอิล-เฟนิล-ยูรีโด (sulfamoyl-phenyl-ureido)ที่มีสูตร (I) ชนิดใหม่ หรือ เกลือหรืออนุพันธ์ซึ่งเป็นที่ยอมรับทางสรีรวิทยาของสารนั้นซึ่งเหมาะสำหรับการบำบัดรักษาการติดเชื้อที่มีสาเหตุโดยโพรโทซัว และโดยเฉพาะโรคมาลาเรียที่ไม่มีอาการแทรกซ้อนหรือรุนแรงที่มีสารเหตุโดยเชื้อ plasmodia
Also published as
SG173171
EP2391601
CN102300844
CA2750967
EA201190031
KR1020110108380
BRPI1007931
AU2010209926
ID051.4424
JP2012516294
PH1/2011/501494
WO/2010/086177
NZ593254
IN1256/MUMNP/2011
IL213996
MX2011007897
UAa201110365
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