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1. WO2004069282 - CONJUGATES OF ENANTIOMER-PURE (4S,8S)- AND (4R,8R)-4-P-BENZYL-8-METHYL-3,6,9-TRIAZA-3N,6N,9N-TRICARBOXYMETHYL-1,11-UNDECANOIC ACID WITH BIOMOLECULES, METHOD FOR THE PRODUCTION THEREOF AND THEIR USE FOR PRODUCING PHARMACEUTICAL AGENTS

Publication Number WO/2004/069282
Publication Date 19.08.2004
International Application No. PCT/EP2003/014922
International Filing Date 22.12.2003
Chapter 2 Demand Filed 25.06.2004
IPC
A61K 51/10 2006.1
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
51Preparations containing radioactive substances for use in therapy or testing in vivo
02characterised by the carrier
04Organic compounds
08Peptides, e.g. proteins
10Antibodies or immunoglobulins; Fragments thereof
CPC
A61K 51/1093
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
51Preparations containing radioactive substances for use in therapy or testing in vivo
02characterised by the carrier ; , i.e. characterised by the agent or material covalently linked or complexing the radioactive nucleus
04Organic compounds
08Peptides, e.g. proteins ; , carriers being peptides, polyamino acids, proteins
10Antibodies or immunoglobulins; Fragments thereof ; , the carrier being an antibody, an immunoglobulin or a fragment thereof, e.g. a camelised human single domain antibody or the Fc fragment of an antibody
1093conjugates with carriers being antibodies
Applicants
  • SCHERING AKTIENGESELLSCHAFT [DE]/[DE]
Inventors
  • LEHMANN, Lutz
  • FRIEBE, Matthias
  • BRUMBY, Thomas
  • SÜLZLE, Detlev
  • PLATZEK, Johannes
Agents
  • TEIPEL, Stephan
Priority Data
103 05 462.604.02.2003DE
Publication Language German (de)
Filing Language German (DE)
Designated States
Title
(DE) KONJUGATE ENANTIOMERENREINER (4S,8S)- UND (4R,8R)-4-P-BENZYL--8-METHYL-3,6,9-TRIAZA-3N,6N,9N-TRICARBOXYMETHYL-1,11-UNDECANDISÄURE MIT BIOMOLEKÜLEN, VERFAHREN ZU DEREN HERSTELLUNG UND VERWENDUNG ZUR HERSTELLUNG PHARMAZEUTISCHER MITTEL
(EN) CONJUGATES OF ENANTIOMER-PURE (4S,8S)- AND (4R,8R)-4-P-BENZYL-8-METHYL-3,6,9-TRIAZA-3N,6N,9N-TRICARBOXYMETHYL-1,11-UNDECANOIC ACID WITH BIOMOLECULES, METHOD FOR THE PRODUCTION THEREOF AND THEIR USE FOR PRODUCING PHARMACEUTICAL AGENTS
(FR) CONJUGUES D'ACIDES (4S,8S)-4-P-BENZYL-8-METHYL-3,6,9-TRIAZA-3N,6N,9N-TRICARBOXYMETHYL-1,11-UNDECANOIQUE ET (4R,8R)-4-P-BENZYL-8-METHYL-3,6,9-TRIAZA-3N,6N,9N-TRICARBOXYMETHYL-1,11-UNDECANOIQUE ENANTIOMERIQUEMENT PURS AVEC DES BIOMOLECULES, PROCEDES DE PRODUCTION DE CES CO
Abstract
(DE) Die Erfindung betrifft enantiomerenreine Konjugate der allgemeinen Formeln (VIIa) und (VIIb) worin A für eine Gruppe -COO- steht und Z und R unterschiedliche Bedeutungen haben, und deren Verwendung.
(EN) The invention relates to enantiomer-pure conjugates of general formulas (VIIa) and (VIIb), wherein A represents a group COO , and Z and R have different meanings. The invention also relates to the use of these conjugates.
(FR) L'invention concerne des conjugués énantiomériquement purs représentés par les formules générales VIIa et VIIb, dans lesquelles A représente un groupe -COO- et Z et R ont des significations différentes, ainsi que leur utilisation.
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