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1. MXMX/a/2007/011769 - PIPERIDINYL SUBSTITUTED CYCLOHEXANE-1,4-DIAMINES

Office Mexico
Application Number MX/a/2007/011769
Application Date 21.09.2007
Publication Number MX/a/2007/011769
Publication Date 27.06.2008
Publication Kind A
IPC
A61K 31/445
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31Medicinal preparations containing organic active ingredients
33Heterocyclic compounds
395having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
435having six-membered rings with one nitrogen as the only ring hetero atom
44Non-condensed pyridines; Hydrogenated derivatives thereof
445Non-condensed piperidines, e.g. piperocaine
A61K 31/454
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31Medicinal preparations containing organic active ingredients
33Heterocyclic compounds
395having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
435having six-membered rings with one nitrogen as the only ring hetero atom
44Non-condensed pyridines; Hydrogenated derivatives thereof
445Non-condensed piperidines, e.g. piperocaine
4523containing further heterocyclic ring systems
454containing a five-membered ring with nitrogen as a ring hetero atom, e.g. pimozide, domperidone
C07D 211/26
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
211Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
04with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
06having no double bonds between ring members or between ring members and non-ring members
08with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
18with substituted hydrocarbon radicals attached to ring carbon atoms
26with hydrocarbon radicals, substituted by nitrogen atoms
C07D 401/02
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
401Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
02containing two hetero rings
Applicants JOHNSON&JOHNSON.*
Inventors CONNOLLY, Peter J.
MIDDLETON, Steven A.
CHIU, George
LI, Shengjian
PULITO, Virginia L.
LIU, Jingchun
Agents HERIBERTO RAUL LOPEZ PADILLA.*
Priority Data 60/664,302 22.03.2005 US
Title
(EN) PIPERIDINYL SUBSTITUTED CYCLOHEXANE-1,4-DIAMINES
(ES) CICLOHEXANO-1,4-DIAMINAS SUSTITUIDAS CON PIPERIDINILO
Abstract
(EN)
The present invention relates to piperidine substituted cyclohexane-1,4-diamine compounds of Formula (I) and pharmaceutically acceptable forms thereof, as a1a/a1d adrenoreceptor modulators for the treatment of benign prostatic hypertrophy and lower urinary tract symptoms. The present invention also relates to pharmaceutical compositions comprising said new compounds, new processes to prepare these new compounds and new uses as a medicine as well as method of treatments.

(ES)
La presente invención se refiere a compuestos ciclohexan-1,4-diamina piperidin sustituidos de fórmula (I) (ver fórmula (I)) y formas farmacéuticamente aceptables de los mismos, como moduladores del adrenorreceptor de ala/ald para el tratamiento de hipertrofia prostática benigna y síntomas del tracto urinario inferior;la presente invención también se refiere a composiciones farmacéuticas que comprenden dichos nuevos compuestos, a nuevos procedimientos para preparar estos nuevos compuestos y a nuevos usos como medicina asícomo a métodos de tratamiento.