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1. KR1020190011240 - 비스페놀 유도체 및 안드로겐 수용체 활성도 조절제로서의 이의 용도

Office Republic of Korea
Application Number 1020187033112
Application Date 18.04.2017
Publication Number 1020190011240
Publication Date 01.02.2019
Publication Kind A
IPC
C07C 43/23
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
CACYCLIC OR CARBOCYCLIC COMPOUNDS
43Ethers; Compounds having groups, groups or groups
02Ethers
20having an ether-oxygen atom bound to a carbon atom of a six-membered aromatic ring
23containing hydroxy or O-metal groups
A61K 31/09
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31Medicinal preparations containing organic active ingredients
075Ethers or acetals
085having an ether linkage to aromatic ring nuclear carbon
09having two or more such linkages
A61K 31/10
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31Medicinal preparations containing organic active ingredients
095Sulfur, selenium or tellurium compounds, e.g. thiols
10Sulfides; Sulfoxides; Sulfones
A61K 31/4164
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31Medicinal preparations containing organic active ingredients
33Heterocyclic compounds
395having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
41having five-membered rings with two or more ring hetero atoms, at least one of which is nitrogen, e.g. tetrazole
41641,3-Diazoles
A61K 31/5375
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31Medicinal preparations containing organic active ingredients
33Heterocyclic compounds
395having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
535having six-membered rings with at least one nitrogen and at least one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
53751,4-Oxazines, e.g. morpholine
A61K 45/06
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
45Medicinal preparations containing active ingredients not provided for in groups A61K31/-A61K41/132
06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
Applicants 브리티쉬 콜롬비아 캔써 에이전시 브랜치
더 유니버시티 오브 브리티쉬 콜롬비아
Inventors 안데르센 레이몬드
사다르 마리안느 도로시
지안 쿤종
마우지 나스린 알.
왕 준
바누엘로스 카르멘 아드리아나
양 유-치
Agents 정홍식
김태헌
Priority Data 62/323,196 15.04.2016 US
Title
(KO) 비스페놀 유도체 및 안드로겐 수용체 활성도 조절제로서의 이의 용도
Abstract
(KO)
하기 화학식 I의 구조를 갖는 화합물 또는 이의 약제학적으로 허용 가능한 염, 호변이성질체 또는 입체이성질체가 제공된다: 식 중, R, R, R, R, R, R, R 및 X는, 본 명세서에서 정의된 바와 같다. 안드로겐 수용체 활성도의 조절, 암의 영상 진단 및 치료제를 위한 이러한 화합물의 용도, 그리고 전립선암을 비롯하여 치료를 필요로 하는 대상체의 치료 방법이 또한 제공된다. JPEG pct00178.jpg 52 76 1 2 3 11a 11b 11c 11d