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1. (JP2012513381) HCVのマクロ環状プロテアーゼ阻害剤を製造するための方法および中間体

Office : Japan
Application Number: 2011541509 Application Date: 22.12.2009
Publication Number: 2012513381 Publication Date: 14.06.2012
Grant Number: 5687631 Grant Date: 18.03.2015
Publication Kind : B2
IPC:
C07D 307/00
C07C 231/12
C07D 453/04
C07C 235/40
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
D
HETEROCYCLIC COMPOUNDS
307
Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
C
ACYCLIC OR CARBOCYCLIC COMPOUNDS
231
Preparation of carboxylic acid amides
12
by reactions not involving the formation of carboxamide groups
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
D
HETEROCYCLIC COMPOUNDS
453
Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
02
containing not further condensed quinuclidine ring systems
04
having a quinolyl-4, a substituted quinolyl-4 or a alkylenedioxy-quinolyl-4 radical linked through only one carbon atom, attached in position 2, e.g. quinine
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
C
ACYCLIC OR CARBOCYCLIC COMPOUNDS
235
Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms
40
having carbon atoms of carboxamide groups bound to carbon atoms of rings other than six-membered aromatic rings and singly-bound oxygen atoms bound to the same carbon skeleton
Applicants: ジヤンセン・フアーマシユーチカルズ・インコーポレーテツド
Janssen Pharmaceuticals,Inc.
Inventors: ホルバト,アンドラス
オルメロド,ドミニク・ジヨン
デプレ,ドミニク・ポール・ミシエル
セルペンテイエ,ベロニク
Agents: 特許業務法人小田島特許事務所
Priority Data: 08172691.1 23.12.2008 EP
Title: (JA) HCVのマクロ環状プロテアーゼ阻害剤を製造するための方法および中間体
Abstract:
(JA)

【化1】

本発明は、マクロ環状HCV阻害剤を製造するための中間体の製造において有用なシンコニジン塩、ならびにこの塩を必要とする方法に関する。


Also published as:
AR074863IL213246MXMX/a/2011/006764EP2382198US20110257403CN102264715
RU2011130895CA2745565ES2429013PT2382198MX2011006764US20150080577
KR1020110099048BRPI0923393RU0002588132DK2382198AU2009331530IN1505/MUMNP/2011
RU2016120007WO/2010/072742