JP2019535771 ７Ｈ－ピロロ［２、３－ｄ］ピリミジン化合物の結晶形、塩型並びにその製造方法

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Single Family Member

Include NPL

Office

Japan

Application Number 2019527838

Application Date 23.11.2017

Publication Number 2019535771

Publication Date 12.12.2019

Grant Number 6788114

Grant Date 02.11.2020

Publication Kind B2

IPC

CPC

Applicants 无▲錫▼福祈制▲薬▼有限公司

Inventors 毛魏魏
▲呉▼▲顕▼
郭▲強▼
▲鄭▼学建
廖勇▲剛▼

Agents 特許業務法人謝国際特許商標事務所
特許業務法人雄渾

Priority Data 201611046683.X 23.11.2016 CN

Title

(JA) ７Ｈ－ピロロ［２、３－ｄ］ピリミジン化合物の結晶形、塩型並びにその製造方法

Abstract

(JA)

本発明は、７Ｈ−ピロロ［２、３−ｄ］ピリミジン化合物の結晶形、塩型並びにその製造方法に関し、また、当該結晶形と塩型の、関節炎治療薬の製造における応用にも関する。
【選択図】図１

C	CHEMISTRY; METALLURGY
07	ORGANIC CHEMISTRY
D	HETEROCYCLIC COMPOUNDS
519	Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/ or C07D455/257

A	HUMAN NECESSITIES
61	MEDICAL OR VETERINARY SCIENCE; HYGIENE
K	PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31	Medicinal preparations containing organic active ingredients
33	Heterocyclic compounds
395	having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
495	having six-membered rings with two nitrogen atoms as the only ring hetero atoms, e.g. piperazine
505	Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
519	ortho- or peri-condensed with heterocyclic rings

A	HUMAN NECESSITIES
61	MEDICAL OR VETERINARY SCIENCE; HYGIENE
P	SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
19	Drugs for skeletal disorders
02	for joint disorders, e.g. arthritis, arthrosis

A	HUMAN NECESSITIES
61	MEDICAL OR VETERINARY SCIENCE; HYGIENE
P	SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
29	Non-central analgesic, antipyretic or antiinflammatory agents, e.g antirheumatic agents; Non-steroidal antiinflammatory drugs (NSAIDs)

C	CHEMISTRY; METALLURGY
07	ORGANIC CHEMISTRY
D	HETEROCYCLIC COMPOUNDS
519	Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/ or C07D455/257

C	CHEMISTRY; METALLURGY
07	ORGANIC CHEMISTRY
B	GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
2200	Indexing scheme relating to specific properties of organic compounds
13	Crystalline forms, e.g. polymorphs