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1. (JP2015522618) 5−HT3受容体拮抗薬

Office : Japan
Application Number: 2015523192 Application Date: 16.07.2013
Publication Number: 2015522618 Publication Date: 06.08.2015
Grant Number: 5816400 Grant Date: 02.10.2015
Publication Kind : B2
IPC:
A61K 31/5386
C07D 498/08
A61P 43/00
A61P 25/24
A61P 25/28
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
K
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31
Medicinal preparations containing organic active ingredients
33
Heterocyclic compounds
395
having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins
535
having six-membered rings with at least one nitrogen and at least one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
5375
1,4-Oxazines, e.g. morpholine
5386
spiro-condensed or forming part of bridged ring systems
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
D
HETEROCYCLIC COMPOUNDS
498
Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
02
in which the condensed system contains two hetero rings
08
Bridged systems
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
P
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
43
Drugs for specific purposes, not provided for in groups A61P1/-A61P41/108
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
P
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
25
Drugs for disorders of the nervous system
24
Antidepressants
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
P
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
25
Drugs for disorders of the nervous system
28
for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
Applicants: 武田薬品工業株式会社
Inventors: ヒッチコック、ステファン
モネシャイン、ホルガー
レイチャード、ホリー
スン、フイカイ
菊地 正太
マクリン、トッド
ホプキンス、マリア
Agents: 高島 一
土井 京子
鎌田 光宜
田村 弥栄子
村田 美由紀
小池 順造
當麻 博文
Priority Data: 61/672,709 17.07.2012 US
61/708,521 01.10.2012 US
Title: (JA) 5−HT3受容体拮抗薬
Abstract:
(JA)

本発明は、嘔吐、疼痛、薬物依存症、神経変性及び精神疾患及びGI障害のような5−HT3受容体の阻害により治療可能な疾患の治療に有用な式(I)の5−HT3受容体拮抗薬を提供する。また、上記化合物を含む医薬組成物及び上記化合物を調製するためのプロセスを提供する。

【選択図】なし


Also published as:
CA2879115IL236702DOP2015000009EP2875011EA201590228SG11201500302U
CN104768943NZ704814AU2013290375BR112015001028ID2016/04647MYPI 2015000110
PH1/2015/500085VN42301IN957/DELNP/2015ES2659758EP3312169TH180869
TN2015000018WO/2014/014951