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1. ID2017/04491 - PYRIDINYL AND FUSED PYRIDINYL TRIAZOLONE DERIVATIVES

Office
Indonesia
Application Number P00201506441
Application Date 10.03.2014
Publication Number 2017/04491
Publication Date 28.04.2017
Publication Kind A
IPC
A61K 31/4725
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31Medicinal preparations containing organic active ingredients
33Heterocyclic compounds
395having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
435having six-membered rings with one nitrogen as the only ring hetero atom
47Quinolines; Isoquinolines
472Non-condensed isoquinolines, e.g. papaverine
4725containing further heterocyclic rings
A61P 35/00
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
35Antineoplastic agents
C07D 401/04
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
401Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
02containing two hetero rings
04directly linked by a ring-member-to-ring- member bond
C07D 401/14
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
401Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
14containing three or more hetero rings
C07D 403/14
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
403Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/167
14containing three or more hetero rings
Applicants TAKEDA PHARMACEUTICAL COMPANY LIMITED
Inventors LAWSON, John David
SMITH, Christopher
SABAT, Mark
SCORAH, Nicholas
VU, Phong H.
WANG, Haixia
Agents Prof. Dr. Toeti Heraty N. Roosseno, Cs.
Title
(EN) PYRIDINYL AND FUSED PYRIDINYL TRIAZOLONE DERIVATIVES
(ID) PIRIDINIL DAN TURUNAN PIRIDINIL TRIAZOLON YANG DISATUKAN
Abstract
(EN)
Disclosed are compounds of Formula 1, or pharmaceutically acceptable salts thereof, wherein R

(ID)
Yang diungkapkan adalah senyawa Rumus 1, atau garam daripadanya yang dapat diterima secara farmasi, di mana R1, R2, R3, dan R4 didef inisikan dalam spesifikasi. Pengungkapan ini juga berhubungan dengan bahan dan metode untuk membuat senyawa Rumus 1, dengan komposisi farmasi yang mengandung senyawa tersebut, dan dengan penggunaannya untuk mengobati reaksi hipersensitivitas Tipe I, penyakit autoimun, gangguan inflamasi, kanker, gangguan proliferasi tidak ganas, dan kondisi lain yang berhubungan dengan BTK.