ES2870006 Procedimiento para producir compuestos que tienen actividad inhibidora de la integrasa del HIV

Office

Spain

Application Number 18203589

Application Date 04.08.2011

Publication Number 2870006

Publication Date 26.10.2021

Publication Kind T3

IPC

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Applicants Shionogi & Co., Ltd

Inventors SUMINO, Yukihito
OKAMOTO, Kazuya
MASUI, Moriyasu
YAMADA, Daisuke
IKARASHI, Fumiya

Agents González Peces Gustavo Adolfo

Priority Data 2010175899 05.08.2010 JP
2010277713 14.12.2010 JP

Title

(ES) Procedimiento para producir compuestos que tienen actividad inhibidora de la integrasa del HIV

Abstract

(ES) Un cristal de un compuesto mostrado por la fórmula (U2) o un solvato del mismo: **(Ver fórmula)** (en la que Me es metilo y Bn es bencilo) que tiene máximos en un espectro de difracción de rayos X en polvo en un ángulo de difracción (2θ): 7,3° ± 0,2°, 14,4° ± 0,2°, 16,1° ± 0,2°, 18,4° ± 0,2°, 22,3° ± 0,2° y 23,1° ± 0,2°.

C	CHEMISTRY; METALLURGY
07	ORGANIC CHEMISTRY
D	HETEROCYCLIC COMPOUNDS
498	Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
12	in which the condensed system contains three hetero rings
14	Ortho-condensed systems

C	CHEMISTRY; METALLURGY
07	ORGANIC CHEMISTRY
D	HETEROCYCLIC COMPOUNDS
211	Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
92	with a hetero atom directly attached to the ring nitrogen atom
94	Oxygen atom, e.g. piperidine N-oxide

C	CHEMISTRY; METALLURGY
07	ORGANIC CHEMISTRY
D	HETEROCYCLIC COMPOUNDS
213	Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
02	having three double bonds between ring members or between ring members and non-ring members
04	having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
60	with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
78	Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
79	Acids; Esters
80	in position 3

A	HUMAN NECESSITIES
61	MEDICAL OR VETERINARY SCIENCE; HYGIENE
K	PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
31	Medicinal preparations containing organic active ingredients
33	Heterocyclic compounds
395	having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
535	having six-membered rings with at least one nitrogen and at least one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
5365	ortho- or peri-condensed with heterocyclic ring systems

A	HUMAN NECESSITIES
61	MEDICAL OR VETERINARY SCIENCE; HYGIENE
P	SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
31	Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
12	Antivirals
14	for RNA viruses
18	for HIV

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1. ES2870006 - Procedimiento para producir compuestos que tienen actividad inhibidora de la integrasa del HIV

C	CHEMISTRY; METALLURGY
07	ORGANIC CHEMISTRY
B	GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
2200	Indexing scheme relating to specific properties of organic compounds
13	Crystalline forms, e.g. polymorphs

A	HUMAN NECESSITIES
61	MEDICAL OR VETERINARY SCIENCE; HYGIENE
K	PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31	Medicinal preparations containing organic active ingredients
33	Heterocyclic compounds
395	having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
535	having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
5365	ortho- or peri-condensed with heterocyclic ring systems