PATENTSCOPE will be unavailable a few hours for maintenance reason on Tuesday 19.11.2019 at 4:00 PM CET
Search International and National Patent Collections
Some content of this application is unavailable at the moment.
If this situation persists, please contact us atFeedback&Contact
1. (ES2429013) Procedimientos e intermedios para la preparación de un inhibidor macrocíclico de la proteasa de VHC

Office : Spain
Application Number: 09801447 Application Date: 22.12.2009
Publication Number: 2429013 Publication Date: 12.11.2013
Publication Kind : T3
Prior PCT appl.: Application Number:EP2009067715 ; Publication Number:2010072742 Click to see the data
IPC:
C07D 311/06
C07D 417/04
C07D 453/04
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
D
HETEROCYCLIC COMPOUNDS
311
Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings
02
ortho- or peri-condensed with carbocyclic rings or ring systems
04
Benzo [b] pyrans, not hydrogenated in the carbocyclic ring
06
with oxygen or sulfur atoms directly attached in position 2
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
D
HETEROCYCLIC COMPOUNDS
417
Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/196
02
containing two hetero rings
04
directly linked by a ring-member-to-ring- member bond
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
D
HETEROCYCLIC COMPOUNDS
453
Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
02
containing not further condensed quinuclidine ring systems
04
having a quinolyl-4, a substituted quinolyl-4 or a alkylenedioxy-quinolyl-4 radical linked through only one carbon atom, attached in position 2, e.g. quinine
CPC:
C07C 67/475
C07C 231/12
C07C 235/40
C07C 2601/08
C07D 307/33
C07D 417/04
C07D 453/04
Applicants: Ortho-McNeil-Janssen Pharmaceuticals, Inc.
Janssen Pharmaceuticals, Inc.
Inventors: HORVATH, Andras
ORMEROD, Dominic John
DEPRE, Dominique Paul Michel
CERPENTIER, Véronique
Agents: Lehmann Lehmann María Isabel
Priority Data: 08172691 23.12.2008 EP
Title: (ES) Procedimientos e intermedios para la preparación de un inhibidor macrocíclico de la proteasa de VHC
Abstract:
(EN) The present invention relates to the cinchonidine salt useful in the preparation of intermediates for preparing a macrocyclic HCV inhibitor, as well as processes involving this salt.
(FR) La présente invention porte sur le sel de cinchonidine utile dans la préparation d'intermédiaires pour préparer un inhibiteur macrocyclique du VHC ainsi que sur des procédés utilisant ce sel.
Also published as:
AR074863IL213246MXMX/a/2011/006764EP2382198JP2012513381US20110257403
CN102264715RU2011130895CA2745565PT2382198MX2011006764US20150080577
KR1020110099048BRPI0923393RU0002588132DK2382198AU2009331530IN1505/MUMNP/2011
RU2016120007WO/2010/072742