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1. (EP2379550) PIPERIDINE DERIVATIVES USEFUL AS OREXIN ANTAGONISTS

Office : European Patent Office
Application Number: 09795991 Application Date: 21.12.2009
Publication Number: 2379550 Publication Date: 26.10.2011
Publication Kind : A1
Designated States: AL, AT, BA, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LI, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR
Prior PCT appl.: Application Number:EP2009067658 ; Publication Number: Click to see the data
IPC:
C07D 471/04
A61K 31/4439
A61P 25/00
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
D
HETEROCYCLIC COMPOUNDS
471
Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/-C07D463/251
02
in which the condensed system contains two hetero rings
04
Ortho-condensed systems
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
K
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31
Medicinal preparations containing organic active ingredients
33
Heterocyclic compounds
395
having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins
435
having six-membered rings with one nitrogen as the only ring hetero atom
44
Non-condensed pyridines; Hydrogenated derivatives thereof
4427
containing further heterocyclic ring systems
4439
containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
P
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
25
Drugs for disorders of the nervous system
CPC:
C07D 471/04
Applicants: GLAXO GROUP LTD
Inventors: ALVARO GIUSEPPE
AMANTINI DAVID
Priority Data: 0823467 null
EP2009067658 null
GB20080023467 null
WO2009EP67658 null
2009067658 21.12.2009 EP
0823467 23.12.2008 GB
Title: (DE) ALS OREXINANTAGONISTEN GEEIGNETE PIPERIDINDERIVATE
(EN) PIPERIDINE DERIVATIVES USEFUL AS OREXIN ANTAGONISTS
(FR) DÉRIVÉS DE PIPÉRIDINE POUVANT ÊTRE UTILISÉS EN TANT QU'AGONISTES DE L'OREXINE
Abstract:
(EN) This invention relates to imidazopyridylmethylene substituted piperidine derivatives orexin antagonists and their use as pharmaceuticals.
(FR) La présente invention concerne des dérivés de pipéridine substitués avec de l'imidazopyridylméthylène, qui sont des antagonistes de l'orexine, et leur utilisation comme produits pharmaceutiques.
Also published as:
IL213345MXMX/a/2011/006768SG171745JP2012513442US20110257198CN102325770
CA2748294EA201170884MX2011006768KR1020110096129AU2009331601IN5412/DELNP/2011
BRPI0922904WO/2010/072722