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1. (CA2879115) 5-HT3 RECEPTOR ANTAGONISTS

Office : Canada
Application Number: 2879115 Application Date:
Publication Number: 2879115 Publication Date: 23.01.2014
Publication Kind : A1
Prior PCT appl.: Application Number:PCTUS2013050746 ; Publication Number: Click to see the data
IPC:
C07D 498/08
A61K 31/439
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
D
HETEROCYCLIC COMPOUNDS
498
Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
02
in which the condensed system contains two hetero rings
08
Bridged systems
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
K
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31
Medicinal preparations containing organic active ingredients
33
Heterocyclic compounds
395
having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins
435
having six-membered rings with one nitrogen as the only ring hetero atom
439
the ring forming part of a bridged ring system, e.g. quinuclidine
CPC:
C07D 221/22
C07D 451/12
C07D 453/02
C07D 471/04
C07D 471/08
C07D 498/08
C07D 519/00
A61K 31/19
A61K 31/5386
C07D 401/14
C07D 403/14
C07D 487/14
C07D 498/04
C07C 53/18
C07C 53/40
Applicants: TAKEDA PHARMACEUTICAL COMPANY LIMITED
Inventors:
Priority Data: 61/672,709 17.07.2012 US
61/708,521 01.10.2012 US
Title: (EN) 5-HT3 RECEPTOR ANTAGONISTS
(FR) ANTAGONISTES DU RECEPTEUR 5-HT3
Abstract: front page image
(EN) The present invention provides 5-HT3 receptor antagonists of Formula (I): which are useful for the treatment of diseases treatable by inhibition of 5-HT3 receptor such as emesis, pain, drug addiction, neurodegenerative and psychiatric disorders, and GI disorders. Also provided are pharmaceutical compositions containing such compounds and processes for preparing such compounds.


Also published as:
IL236702DOP2015000009EP2875011EA201590228SG11201500302UCN104768943
JP2015522618NZ704814AU2013290375BR112015001028ID2016/04647MYPI 2015000110
PH1/2015/500085VN42301IN957/DELNP/2015ES2659758EP3312169TH180869
TN2015000018WO/2014/014951